racetamEVIDENCECUSUnscheduled
Fasoracetam
Atypical racetam under investigation for adolescent ADHD. Modulates GABA-B, mGluR, and cholinergic systems.
Dose range10–30mg
Half-life5h
Onset30min
Safety4/5low evidence base
Mechanism of action
Upregulates GABA-B receptors. Modulates mGluR groups II/III. Cholinergic enhancement.
Benefits
ADHD symptoms in mGluR-mutation phenotype
EVIDENCECPediatric trials by Aevi.
Anxiolytic via GABA-B
EVIDENCECAnimal models.
Side effects
- Sedation at high doseuncommonmild
- Headacheuncommonmild
Where to buy
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